| 產(chǎn)品編號(hào) | D58189 |
| 英文名稱 | GSK046 |
| 中文名稱 | |
| 別 名 | iBET-BD2 |
| 克 隆 號(hào) | |
| CAS | 2474876-09-8 |
| 理論分子量 | 414.48 kDa |
| 檢測(cè)分子量 | |
| 保存條件 | Powder: -20℃ for 3 years | In solvent: -80℃ for 1 year |
| 注意事項(xiàng) | This product as supplied is intended for research use only, not for use in human, therapeutic or diagnostic applications. |
| 產(chǎn)品介紹 |
GSK046 is a potent, selective and orally active BD2 bromodomain inhibitor of the BET proteins(IC50s of 264 nM (BRD2 BD2), 98 nM (BRD3 BD2), 49 nM (BRD4 BD2) and 214 nM (BRDT BD2), respectively). It has immunomodulatory activity. |
